SCHEMBL20155116

SCHEMBL20155116

CCn1cc2c(=O)n(C)cc(-c3cc(N)ccc3Nc3ccc(F)cc3F)c2n1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 13/20 0.45
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MAT2A P31153 2/20 0.36
MAPK14 Q16539 2/20 0.36
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155171 0.91 BRD4 (0.43) BRD4MAT2A
SCHEMBL20155659 0.88 BRD4 (0.46) BRD4
SCHEMBL20155427 0.88 BRD4 (0.48) BRD4MAPK14TSHRHSD17B10
SCHEMBL20155652 0.85 BRD4 (0.48) BRD4NPC1RAB9AMAT2AMAPK14
SCHEMBL20155689 0.83 BRD4 (0.54) BRD4
SCHEMBL21904958 0.81 BRD4 (0.66) BRD4
SCHEMBL20155185 0.80 BRD4 (0.42) BRD4MAT2A
SCHEMBL20155619 0.79 BRD4 (0.46) BRD4
SCHEMBL20155737 0.79 BRD4 (0.47) BRD4MAT2A
SCHEMBL20155644 0.78 BRD4 (0.45) BRD4MAPK14TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed