SCHEMBL20155659

SCHEMBL20155659

Cn1cc(-c2cc(N)ccc2Nc2ccc(F)cc2F)c2nn(Cc3ccccc3)cc2c1=O

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 15/20 0.46
THRB P10828 1/20 0.36
MEN1 O00255 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CREBBP Q92793 1/20 0.36
BRD2 P25440 1/20 0.35
ADORA3 P0DMS8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155116 0.88 BRD4 (0.45) BRD4
SCHEMBL20155113 0.85 BRD4 (0.48) BRD4THRBMEN1HTTKMT2A
SCHEMBL20155427 0.84 BRD4 (0.48) BRD4
SCHEMBL20155171 0.81 BRD4 (0.43) BRD4CREBBPBRD2
SCHEMBL21904958 0.81 BRD4 (0.66) BRD4
SCHEMBL20155185 0.78 BRD4 (0.42) BRD4
SCHEMBL20155737 0.77 BRD4 (0.47) BRD4
SCHEMBL20155619 0.76 BRD4 (0.46) BRD4
SCHEMBL20155644 0.74 BRD4 (0.45) BRD4
SCHEMBL20155652 0.74 BRD4 (0.48) BRD4BRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed