SCHEMBL20155320

SCHEMBL20155320

Cc1cc(CO)ccc1Oc1ccc(F)cc1F

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.43
CYP4F2 P78329 1/20 0.42
CYP4A11 Q02928 1/20 0.42
CARM1 Q86X55 2/20 0.41
PRMT6 Q96LA8 2/20 0.41
TRPA1 O75762 3/20 0.40
SLC6A4 P31645 1/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
EPAS1 Q99814 1/20 0.39
HSPB1 P04792 1/20 0.38
EP300 Q09472 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10603411 0.85 TTR (0.47) CYP4F2CYP4A11CARM1PRMT6
SCHEMBL20155323 0.84 SLC6A4 (0.43) BRD4CARM1PRMT6TRPA1SLC6A4
SCHEMBL15068243 0.83 EPAS1 (0.52) BRD4CYP4F2CYP4A11TRPA1EPAS1
SCHEMBL20160312 0.79 BRD4 (0.58) BRD4PTGS1PTGS2EPAS1EP300
SCHEMBL20160228 0.76 BRD4 (0.49) BRD4TRPA1SLC6A4HSPB1
SCHEMBL20160295 0.76 EPAS1 (0.44) TRPA1SLC6A4EPAS1HSPB1
SCHEMBL14656214 0.76 TTR (0.51) CYP4F2CYP4A11CARM1PRMT6HSPB1
SCHEMBL31073743 0.76 HSPB1 (0.38) BRD4CYP4F2CYP4A11CARM1PRMT6
SCHEMBL4439280 0.75 SLC6A4 (0.53) SLC6A4PTGS1PTGS2
SCHEMBL10456772 0.75 TRPA1 (0.56) TRPA1EPAS1HSPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed