SCHEMBL20155323

SCHEMBL20155323

Cc1cc(CBr)ccc1Oc1ccc(F)cc1F

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.43
TRPA1 O75762 7/20 0.40
EPAS1 Q99814 1/20 0.39
HSPB1 P04792 2/20 0.38
CARM1 Q86X55 2/20 0.38
PRMT6 Q96LA8 2/20 0.38
BRD4 O60885 3/20 0.38
EP300 Q09472 2/20 0.38
SLC6A2 P23975 2/20 0.37
SLC6A3 Q01959 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155320 0.84 BRD4 (0.43) SLC6A4TRPA1EPAS1HSPB1CARM1
SCHEMBL15067971 0.83 EPAS1 (0.52) TRPA1EPAS1HSPB1CARM1PRMT6
SCHEMBL30444289 0.83 EPAS1 (0.52) TRPA1EPAS1HSPB1CARM1PRMT6
SCHEMBL20160295 0.79 EPAS1 (0.44) SLC6A4TRPA1EPAS1HSPB1
SCHEMBL20160312 0.79 BRD4 (0.58) EPAS1BRD4EP300
SCHEMBL20160228 0.76 BRD4 (0.49) SLC6A4TRPA1HSPB1BRD4SLC6A2
SCHEMBL4439280 0.75 SLC6A4 (0.53) SLC6A4SLC6A2SLC6A3
SCHEMBL10456772 0.75 TRPA1 (0.56) TRPA1EPAS1HSPB1
SCHEMBL9560643 0.75 HSPB1 (0.43) SLC6A4TRPA1HSPB1SLC6A2SLC6A3
SCHEMBL20155430 0.74 TRPA1 (0.45) SLC6A4TRPA1EPAS1HSPB1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed