SCHEMBL20155393

SCHEMBL20155393

CC1(C)OB(c2cc(N)ccc2Oc2ccc(Cl)cc2C#N)OC1(C)C

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
USP2 O75604 1/20 0.42
SLC22A12 Q96S37 10/20 0.36
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
PGGT1B P53609 1/20 0.35
MEN1 O00255 2/20 0.34
HPGD P15428 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C19 P33261 1/20 0.34
NOS2 P35228 1/20 0.34
EGFR P00533 2/20 0.34
SCN9A Q15858 2/20 0.32
SYK P43405 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155469 0.86 KDM4E (0.42) KDM4EALDH1A1USP2SLC22A12
SCHEMBL20155409 0.82 SLC6A2 (0.39) ALDH1A1HPGDEGFRSCN9A
SCHEMBL20155354 0.80 MAPT (0.44) KDM4EALDH1A1MEN1HPGDKMT2A
SCHEMBL18000582 0.79 KDM4E (0.44) KDM4EALDH1A1USP2MEN1HPGD
SCHEMBL28688126 0.79 KDM4E (0.59) KDM4EALDH1A1USP2SLC22A12FNTA
SCHEMBL15069404 0.77 AR (0.39) KDM4EALDH1A1USP2MEN1KMT2A
SCHEMBL13183400 0.77 VCAM1 (0.38) KDM4EALDH1A1MEN1HPGDKMT2A
SCHEMBL11971323 0.77 GPR35 (0.36) KDM4EALDH1A1SLC22A12NOS2EGFR
SCHEMBL30722717 0.77 GPR35 (0.36) KDM4EALDH1A1SLC22A12NOS2EGFR
SCHEMBL20155416 0.75 SLC6A2 (0.40) ALDH1A1HPGDMAPTEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed