SCHEMBL20155400

SCHEMBL20155400

Clc1nccc2nn(C3CC3)cc12

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 4/20 0.39
LRRK2 Q5S007 2/20 0.36
JAK2 O60674 1/20 0.34
TYK2 P29597 1/20 0.34
PTPN11 Q06124 1/20 0.32
LMNA P02545 1/20 0.31
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31
APEX1 P27695 1/20 0.31
MAPK1 P28482 1/20 0.31
PMP22 Q01453 1/20 0.31
CYP2D6 P10635 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155612 0.75 LMNA (0.34) PDE4DJAK2TYK2LMNACYP3A4
SCHEMBL26921636 0.72 PTPN11 (0.35) PDE4DLRRK2PTPN11
SCHEMBL17873844 0.72 ADORA2A (0.40) PTPN11LMNACYP3A4MAPTAPEX1
SCHEMBL29993671 0.71 LRRK2 (0.34) PDE4DLRRK2PTPN11
SCHEMBL24035856 0.68 ACACB (0.34) LMNACYP3A4MAPTAPEX1MAPK1
SCHEMBL20155347 0.68 MAT2A (0.38) PDE4DPTPN11LMNACYP3A4MAPT
SCHEMBL2596927 0.67 PDE4D (0.39) PDE4D
SCHEMBL2077005 0.66 ABL1 (0.46) PDE4DLRRK2
SCHEMBL6119305 0.66 JAK2 (0.56) PDE4DJAK2TYK2LMNACYP3A4
SCHEMBL2075692 0.65 ABL1 (0.48) LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed