SCHEMBL20155447

SCHEMBL20155447

CC1(C)OB(c2cc(N)ccc2Oc2ccc(C#N)cn2)OC1(C)C

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.42
ALOX5AP P20292 3/20 0.39
FEN1 P39748 3/20 0.39
KEAP1 Q14145 1/20 0.33
OPRM1 P35372 1/20 0.33
LIPE Q05469 7/20 0.32
KDM4E B2RXH2 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
DGAT1 O75907 1/20 0.32
EGFR P00533 1/20 0.32
GABRA5 P31644 1/20 0.31
FPR2 P25090 1/20 0.31
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15069404 0.82 AR (0.39) PDE4BKDM4EMEN1KMT2AUSP2
SCHEMBL20155520 0.77 KEAP1 (0.46) PDE4BALOX5APFEN1KEAP1OPRM1
SCHEMBL20155450 0.74 ALOX5AP (0.45) PDE4BALOX5APFEN1KEAP1OPRM1
SCHEMBL2527256 0.73 PDE4B (0.52) PDE4BOPRM1LIPEKDM4EALDH1A1
SCHEMBL20155393 0.73 KDM4E (0.42) KDM4EMEN1KMT2AUSP2ALDH1A1
SCHEMBL20155469 0.73 KDM4E (0.42) KDM4EUSP2ALDH1A1
SCHEMBL18605502 0.71 ALDH1A1 (0.41) KDM4EMEN1KMT2AUSP2ALDH1A1
SCHEMBL15328685 0.71 BRD4 (0.40) MEN1KMT2AALDH1A1
SCHEMBL30083309 0.70 AR (0.42) KDM4EUSP2ALDH1A1EGFR
SCHEMBL1303766 0.70 AR (0.42) KDM4EUSP2ALDH1A1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed