SCHEMBL20155472

SCHEMBL20155472

CN/C=C1\C(=N)C(c2cc(N)ccc2Oc2ccc(C#N)cc2)=CN(C)C1=O

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 4/20 0.35
BRD4 O60885 9/20 0.34
ESRRA P11474 1/20 0.31
PLA2G7 Q13093 1/20 0.30
AR P10275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155487 0.89 BRD4 (0.33) SCN9ABRD4
SCHEMBL20155356 0.88 ALDH1A1 (0.34) BRD4
SCHEMBL20155097 0.86 BRD4 (0.37) BRD4PLA2G7
SCHEMBL20155005 0.84 BRD4 (0.54) BRD4PLA2G7
SCHEMBL20155475 0.82 BRD4 (0.41) BRD4PLA2G7
SCHEMBL20155692 0.78 SLC6A2 (0.34) SCN9ABRD4
SCHEMBL20155007 0.78 SLC6A2 (0.35) BRD4
SCHEMBL20155530 0.74 BRD4 (0.37) BRD4
SCHEMBL20155038 0.72 BRD4 (0.42) BRD4
SCHEMBL20155531 0.70 BRD4 (0.41) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed