SCHEMBL20155565

SCHEMBL20155565

CN(C)CCn1cc2c(=O)[nH]cc(Br)c2n1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.37
KDM4A O75164 2/20 0.32
KDM4B O94953 2/20 0.32
KDM5C P41229 2/20 0.32
KDM5B Q9UGL1 2/20 0.32
DAO P14920 1/20 0.32
KAT2B Q92831 2/20 0.32
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
TOP2A P11388 1/20 0.30
KDM4E B2RXH2 1/20 0.30
TERT O14746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155529 0.77 CNR2 (0.40) CNR2KAT2BTOP2AKDM4ETERT
SCHEMBL20155563 0.73 CNR2 (0.42) CNR2KDM4AKDM4BKDM5CKDM5B
SCHEMBL20155109 0.72 ADORA3 (0.56) DAOKDM4E
SCHEMBL20155615 0.69 GSK3B (0.34) KDM4E
SCHEMBL20155724 0.69 GSK3B (0.32)
SCHEMBL20155157 0.69 GSK3B (0.30)
SCHEMBL20155732 0.66 GSK3B (0.30)
SCHEMBL20155126 0.65 PDE4D (0.34) PDE4D
SCHEMBL28549245 0.65 CYP2D6 (0.35)
SCHEMBL17870698 0.64 PDE4A (0.40) DAOPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed