SCHEMBL20155637

SCHEMBL20155637

CCSCc1ccc(Nc2ccc(F)cc2F)c(C2=CN(C)C(=O)/C(=C/NC)C2=N)c1

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.36
ALDH1A1 P00352 1/20 0.32
MAP2K2 P36507 1/20 0.31
MAP2K1 Q02750 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155590 0.83 MAPK14 (0.36) BRD4ALDH1A1MAP2K2MAP2K1
SCHEMBL20155650 0.78 AKT1 (0.31) BRD4
SCHEMBL20155583 0.78 BRD4 (0.36) BRD4
SCHEMBL20155138 0.76 MAPK14 (0.36) BRD4ALDH1A1
SCHEMBL20155643 0.75 BRD4 (0.35) BRD4ALDH1A1
SCHEMBL20155635 0.75 MAPK14 (0.33) BRD4MAP2K2MAP2K1
SCHEMBL20155186 0.75 TDO2 (0.31)
SCHEMBL20155584 0.75 BRD4 (0.43) BRD4
SCHEMBL20155748 0.74 MAPK14 (0.34) BRD4
SCHEMBL20155483 0.72 MAPK14 (0.37) BRD4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed