SCHEMBL20155728

SCHEMBL20155728

Cn1nc2c(-c3cc(N)ccc3Nc3ccc(Cl)cc3F)cn(C)c(=O)c2n1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 6/20 0.43
NUDT1 P36639 1/20 0.35
EIF2AK3 Q9NZJ5 1/20 0.35
TAS2R14 Q9NYV8 1/20 0.34
MAP2K1 Q02750 5/20 0.33
MAP2K2 P36507 3/20 0.33
TRPM5 Q9NZQ8 1/20 0.33
TSHR P16473 1/20 0.32
TGFBR1 P36897 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155630 0.86 BPTF (0.40) BRD4
SCHEMBL20155737 0.86 BRD4 (0.47) BRD4NUDT1EIF2AK3TAS2R14MAP2K1
SCHEMBL20155506 0.84 BRD4 (0.43) BRD4MAP2K1
SCHEMBL20155171 0.83 BRD4 (0.43) BRD4TGFBR1
SCHEMBL20155107 0.82 BRD4 (0.45) BRD4
SCHEMBL20155427 0.76 BRD4 (0.48) BRD4TSHR
SCHEMBL20155510 0.75 BRD4 (0.47) BRD4
SCHEMBL20155185 0.73 BRD4 (0.42) BRD4
SCHEMBL20155116 0.73 BRD4 (0.45) BRD4TSHR
SCHEMBL20155149 0.71 BRD4 (0.46) BRD4MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed