SCHEMBL20156241

SCHEMBL20156241

CCOC(=O)/C(=C/NCCC1(C)OCCO1)C(=N)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
CYP2D6 P10635 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 3/20 0.34
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
GLO1 Q04760 1/20 0.33
GAA P10253 2/20 0.31
MAPT P10636 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20156326 0.87 ALDH1A1 (0.42) ALDH1A1CYP2D6SMN1; SMN2NPSR1KDM4E
SCHEMBL20156038 0.81 ALDH1A1 (0.36) ALDH1A1CYP2D6SMN1; SMN2GLO1
SCHEMBL20156005 0.80 ALDH1A1 (0.33) ALDH1A1CYP2D6SMN1; SMN2GLO1
SCHEMBL20156244 0.79 CYP2D6 (0.44) ALDH1A1CYP2D6SMN1; SMN2NPSR1KDM4E
SCHEMBL20156293 0.69 KMT2A (0.30)
SCHEMBL13958022 0.67 NPSR1 (0.43) ALDH1A1CYP2D6SMN1; SMN2NPSR1KDM4E
SCHEMBL14391944 0.67 NPSR1 (0.43) ALDH1A1CYP2D6SMN1; SMN2NPSR1KDM4E
SCHEMBL20156243 0.66 MAPT (0.41) CYP2D6NPSR1KDM4EMAPT
SCHEMBL20156072 0.65
SCHEMBL19403663 0.64 HDAC4 (0.41) ALDH1A1NPSR1GLO1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089358-A1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed