Lysine

Lysine

SCHEMBL2015695

C[C@@H](OC(=O)CN)[C@H](NP(=O)(O)O)C(=O)O.NCCCC[C@H](N)C(=O)O

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPARDPTGS1PTGS2dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Lysine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GSR P00390 1/20 0.48
THRB P10828 1/20 0.37
OTC P00480 1/20 0.36
BHMT Q93088 1/20 0.33
ARG1 P05089 3/20 0.33
ARG2 P78540 3/20 0.33
NOS3 P29474 2/20 0.33
NOS1 P29475 2/20 0.33
NOS2 P35228 2/20 0.33
GNAI3 P08754 1/20 0.33
GNAO1 P09471 1/20 0.33
GNAI1 P63096 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
POLB P06746 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lysine SCHEMBL2015699 0.81 GSR (0.51) GSRTHRBOTCARG1ARG2
Lysine SCHEMBL27494734 0.73 GSR (0.77) GSROTCARG1ARG2POLB
Lysine SCHEMBL11803679 0.72 GSR (0.83) GSROTCARG1ARG2POLB
Lysine SCHEMBL1446119 0.72 GSR (0.83) GSROTCARG1ARG2POLB
Lysine SCHEMBL103555 0.72 GSR (0.83) GSROTCARG1ARG2POLB
Lysine SCHEMBL1825922 0.72 GSR (0.83) GSROTCARG1ARG2POLB
Lysine SCHEMBL31708395 0.72 GSR (0.69) GSROTCARG1ARG2NOS3
Lysine SCHEMBL29050532 0.71 GSR (0.74) GSROTCARG1ARG2POLB
Lysine SCHEMBL1666689 0.71 GSR (0.74) GSROTCARG1ARG2POLB
Lysine SCHEMBL11671036 0.71 GSR (0.80) GSROTCARG1ARG2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8244484-B2 Proteome epitope tags and methods of use thereof in protein modification analysis EMD MILLIPORE CORPORATION (US) 2012-08-14 US disclosed
US-7964362-B2 Proteome epitope tags and methods of use thereof in protein modification analysis MILLIPORE CORPORATION (US) 2011-06-21 US disclosed
US-20100331200-A1 POST TRANSLATIONAL MODIFICATION PATTERN ANALYSIS MILLIPORE CORPORATION 2010-12-30 US disclosed
US-20100184613-A1 Proteome Epitope Tags and Methods of Use Thereof in Protein Modification Analysis MILLIPORE CORPORATION (US) 2010-07-22 US disclosed
US-7618788-B2 Proteome epitope tags and methods of use thereof in protein modification analysis MILLIPORE CORPORATION (US) 2009-11-17 US disclosed
US-20090023157-A1 Proteome epitope tags and methods of use thereof in protein modification analysis EMD MILLIPORE CORPORATION 2009-01-22 US disclosed
US-7460960-B2 Proteome epitope tags and methods of use thereof in protein modification analysis EPITOME BIOSYSTEMS, INC. (US) 2008-12-02 US disclosed
WO-2007123708-A2 POST TRANSLATIONAL MODIFICATION PATTERN ANALYSIS EPITOME BIOSYSTEMS, INC. (US) 2007-11-01 WO disclosed
EP-1683065-A2 PROTEOME EPITOPE TAGS AND METHODS OF USE THEREOF IN PROTEIN MODIFICATION ANALYSIS Epitome Biosystems, Inc. (US) 2006-07-26 EP disclosed
US-20060014212-A1 Proteome epitope tags and methods of use thereof in protein modification analysis EPITOME BIOSYSTEMS, INC. (US) 2006-01-19 US disclosed
WO-2005078453-A2 PROTEOME EPITOPE TAGS AND METHODS OF USE THEREOF IN PROTEIN MODIFICATION ANALYSIS EPITOME BIOSYSTEMS INC. (US) 2005-08-25 WO disclosed
WO-2005050223-A2 PROTEOME EPITOPE TAGS AND METHODS OF USE THEREOF IN PROTEIN MODIFICATION ANALYSIS EPITOME BIOSYSTEMS INC. (US) 2005-06-02 WO disclosed
US-20050069911-A1 Using peptide probes to for high sensitivity/accuracy in detection quantitation of target proteins; biosignatures and disease diagnosis ENGENEOS, INC. (US) 2005-03-31 US disclosed
US-20040180380-A1 Proteome epitope tags and methods of use thereof in protein modification analysis ENGENEOS, INC. 2004-09-16 US disclosed