SCHEMBL20157244

SCHEMBL20157244

N#Cc1ccccc1N1CCC2CNC(C2)C1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 3/20 0.43
GRM5 P41594 1/20 0.42
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 1/20 0.40
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
CYP3A4 P08684 1/20 0.36
DRD4 P21917 2/20 0.36
DRD2 P14416 1/20 0.34
GRM2 Q14416 1/20 0.34
CHRM4 P08173 1/20 0.34
KDM1A O60341 1/20 0.34
AR P10275 1/20 0.34
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
CDC42BPB Q9Y5S2 1/20 0.34
C5AR1 P21730 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157269 0.81 ALDH1A1 (0.36) KDM4EALDH1A1CHRNB2CHRNA4
SCHEMBL20140205 0.77 GRM1 (0.47) GRM1GRM5KDM4EDRD4DRD2
SCHEMBL12835705 0.75 DPP4 (0.47) GRM1GRM5KDM4EALDH1A1
SCHEMBL20129683 0.75 DPP4 (0.47) GRM1GRM5KDM4EALDH1A1
SCHEMBL20139200 0.75 GRM1 (0.43) GRM1GRM5KDM4EALDH1A1CHRNB2
SCHEMBL23702949 0.74 AR (0.55) GRM1GRM5KDM4EALDH1A1CYP3A4
Hydrochloric Acid SCHEMBL1514528 0.74 DPP4 (0.47) GRM1GRM5KDM4EALDH1A1
SCHEMBL23708047 0.74 AR (0.55) GRM1GRM5KDM4EALDH1A1CYP3A4
Hydrochloric Acid SCHEMBL1514285 0.74 DPP4 (0.47) GRM1GRM5KDM4EALDH1A1
SCHEMBL23708107 0.74 AR (0.55) GRM1GRM5KDM4EALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed