SCHEMBL20157342

SCHEMBL20157342

CCS(=O)(=O)Cc1ccc(C(=O)c2ccc(C)cc2)c(Br)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.43
MAPT P10636 5/20 0.43
KMT2A Q03164 3/20 0.41
HTT P42858 3/20 0.40
RAB9A P51151 1/20 0.40
NPC1 O15118 1/20 0.40
MAPK1 P28482 1/20 0.40
ALDH1A1 P00352 3/20 0.40
LMNA P02545 1/20 0.40
CA2 P00918 1/20 0.38
AKR1C3 P42330 1/20 0.38
KDM5A P29375 1/20 0.38
GAA P10253 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RXRA P19793 1/20 0.36
C5AR1 P21730 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21362472 0.89 SRD5A2 (0.43) SRD5A2MAPTKMT2AHTTRAB9A
SCHEMBL20157579 0.88 TP53 (0.38) MAPTKMT2AHTTMAPK1ALDH1A1
SCHEMBL20157815 0.88 KMT2A (0.40) SRD5A2MAPTKMT2ARAB9ANPC1
SCHEMBL20157951 0.88 MAPT (0.47) SRD5A2MAPTHTTRAB9ANPC1
SCHEMBL20157411 0.86 NPC1 (0.48) MAPTKMT2AHTTRAB9ANPC1
SCHEMBL21351995 0.85 CCR9 (0.47) MAPTKMT2AHTTRAB9ANPC1
SCHEMBL20157973 0.85 SRD5A2 (0.42) SRD5A2MAPTHTTRAB9ANPC1
SCHEMBL20157469 0.85 POLB (0.47) SRD5A2MAPTKMT2AHTTRAB9A
SCHEMBL21362746 0.85 TAS1R3 (0.35) SRD5A2MAPTHTTCA2AKR1C3
SCHEMBL20158071 0.83 KMT2A (0.36) MAPTKMT2AHTTNPC1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed