SCHEMBL21362472

SCHEMBL21362472

CCS(=O)(=O)Cc1ccc(Br)c(C(=O)c2ccc(C)cc2)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.43
MAPT P10636 5/20 0.43
KMT2A Q03164 4/20 0.41
HTT P42858 3/20 0.40
RAB9A P51151 1/20 0.40
NPC1 O15118 1/20 0.40
MAPK1 P28482 1/20 0.40
ALDH1A1 P00352 3/20 0.40
LMNA P02545 1/20 0.40
CA2 P00918 1/20 0.38
AKR1C3 P42330 1/20 0.38
KDM5A P29375 1/20 0.38
GAA P10253 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RXRA P19793 1/20 0.36
C5AR1 P21730 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157342 0.89 SRD5A2 (0.43) SRD5A2MAPTKMT2AHTTRAB9A
SCHEMBL20157851 0.88 THRB (0.38) MAPTKMT2AHTTALDH1A1LMNA
SCHEMBL20157429 0.81 SRD5A2 (0.49) SRD5A2MAPTKMT2AHTTRAB9A
SCHEMBL24199841 0.79 MAPT (0.51) SRD5A2MAPTKMT2AHTTRAB9A
SCHEMBL20157997 0.78 MAPT (0.40) SRD5A2MAPTKMT2AHTTRAB9A
SCHEMBL20157430 0.77 MAPT (0.60) SRD5A2MAPTHTTRAB9ANPC1
SCHEMBL20157815 0.77 KMT2A (0.40) SRD5A2MAPTKMT2ARAB9ANPC1
SCHEMBL20157579 0.77 TP53 (0.38) MAPTKMT2AHTTMAPK1ALDH1A1
SCHEMBL20157951 0.77 MAPT (0.47) SRD5A2MAPTHTTRAB9ANPC1
SCHEMBL20158141 0.76 MAPT (0.41) MAPTHTTNPC1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed