SCHEMBL20157480

SCHEMBL20157480

COc1cc(C(=O)c2ccc(C(Br)Br)cc2Br)ccc1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
CYP1A2 P05177 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
HPGD P15428 4/20 0.41
CYP2D6 P10635 1/20 0.41
SLC22A6 Q4U2R8 1/20 0.40
SLC22A8 Q8TCC7 1/20 0.40
NPC1 O15118 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
KMT2A Q03164 1/20 0.39
MAPT P10636 3/20 0.38
GAA P10253 2/20 0.38
HTT P42858 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PDF Q9HBH1 1/20 0.37
LCK P06239 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21362792 0.91 ALDH1A1 (0.44) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL20157647 0.86 ALDH1A1 (0.44) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL21550011 0.86 ALDH1A1 (0.44) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL20157483 0.84 ALDH1A1 (0.50) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL20158085 0.84 HTT (0.50) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL21352037 0.81 NPC1 (0.54) ALDH1A1CYP1A2CYP2C19CYP3A4TSHR
SCHEMBL21362793 0.80 PKM (0.49) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL20157609 0.80 ALDH1A1 (0.46) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL21564711 0.78 ALDH1A1 (0.43) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL21352048 0.75 LCK (0.38) ALDH1A1NPC1KMT2AMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed