SCHEMBL21362793

SCHEMBL21362793

CCc1ccc(C(=O)c2ccc(C)c(OC)c2)c(Br)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.49
ALDH1A1 P00352 2/20 0.46
ACHE P22303 3/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
HPGD P15428 2/20 0.41
HSD17B2 P37059 1/20 0.41
CYP2D6 P10635 1/20 0.41
SLC22A6 Q4U2R8 1/20 0.40
SLC22A8 Q8TCC7 1/20 0.40
NPC1 O15118 2/20 0.40
BCHE P06276 2/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
RAB9A P51151 1/20 0.39
MAPT P10636 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157609 0.90 ALDH1A1 (0.46) PKMALDH1A1ACHECYP1A2CYP2C19
SCHEMBL20157485 0.87 ALDH1A1 (0.41) PKMALDH1A1ACHECYP1A2CYP2C19
SCHEMBL21564843 0.86 ALDH1A1 (0.44) ALDH1A1ACHECYP1A2CYP2C19CYP3A4
SCHEMBL20158058 0.84 ALDH1A1 (0.41) PKMALDH1A1ACHECYP1A2CYP2C19
SCHEMBL21362509 0.84 MAPT (0.45) PKMALDH1A1ACHECYP1A2CYP2C19
SCHEMBL20157483 0.84 ALDH1A1 (0.50) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL24199867 0.82 HTT (0.45) PKMALDH1A1ACHECYP1A2CYP2C19
SCHEMBL20157480 0.80 ALDH1A1 (0.46) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL21362792 0.79 ALDH1A1 (0.44) PKMALDH1A1CYP1A2CYP2C19CYP3A4
SCHEMBL20158011 0.77 CA12 (0.38) ALDH1A1ACHECYP1A2CYP2C19HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed