SCHEMBL20157513

SCHEMBL20157513

COc1cc(F)ccc1C(=O)c1ccc(CBr)cc1CBr

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
RAB9A P51151 1/20 0.46
FFAR4 Q5NUL3 3/20 0.41
FFAR1 O14842 1/20 0.41
LPAR1 Q92633 1/20 0.38
LPAR5 Q9H1C0 1/20 0.38
PYGL P06737 1/20 0.37
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.36
CTSL P07711 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
CLK1 P49759 1/20 0.36
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157512 0.87 NPC1 (0.46) NPC1SMN1; SMN2RAB9AFFAR4FFAR1
SCHEMBL20158051 0.85 SMN1; SMN2 (0.39) NPC1SMN1; SMN2RAB9AFFAR4FFAR1
SCHEMBL27709578 0.81 NPC1 (0.51) NPC1SMN1; SMN2RAB9AFFAR4FFAR1
SCHEMBL20157850 0.76 MAPT (0.39) NPC1SMN1; SMN2RAB9AFFAR4FFAR1
SCHEMBL21362429 0.75 SMN1; SMN2 (0.41) NPC1SMN1; SMN2RAB9AFFAR4FFAR1
SCHEMBL4440969 0.74 CES2 (0.39) NPC1SMN1; SMN2RAB9AKMT2AMEN1
SCHEMBL1121702 0.74 NPC1 (0.55) NPC1SMN1; SMN2RAB9AFFAR4FFAR1
SCHEMBL7703503 0.74 FFAR4 (0.45) NPC1SMN1; SMN2RAB9AFFAR4ALDH1A1
SCHEMBL3916859 0.73 MAPT (0.54) NPC1SMN1; SMN2RAB9AKMT2AALDH1A1
SCHEMBL18310131 0.72 SMN1; SMN2 (0.47) NPC1SMN1; SMN2RAB9AKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed