SCHEMBL20157559

SCHEMBL20157559

Bc1cnc(N)cc1C#N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1A1 P48729 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
PIK3CA P42336 1/20 0.36
PIK3CD O00329 1/20 0.36
NOS3 P29474 2/20 0.35
NOS1 P29475 2/20 0.35
NOS2 P35228 2/20 0.35
ALOX5AP P20292 3/20 0.33
FEN1 P39748 3/20 0.33
HTT P42858 1/20 0.33
PDPK1 O15530 1/20 0.33
KDR P35968 2/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
ABL1 P00519 1/20 0.32
KDM4E B2RXH2 2/20 0.32
KHK P50053 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
GSK3B P49841 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21011621 0.83 CSNK1A1 (0.41) CSNK1A1CLK4PIK3CAPIK3CDNOS3
SCHEMBL16668748 0.80 CSNK1A1 (0.45) CSNK1A1CLK4PIK3CAPIK3CDNOS3
SCHEMBL11486802 0.78 PIK3CD (0.42) CSNK1A1CLK4PIK3CAPIK3CDNOS3
SCHEMBL18031200 0.75 NOS3 (0.56) CSNK1A1CLK4PIK3CAPIK3CDNOS3
SCHEMBL1815383 0.75 XDH (0.40) CSNK1A1CLK4PIK3CAPIK3CDNOS3
SCHEMBL23908930 0.75 XDH (0.39) CSNK1A1CLK4PIK3CAPIK3CDNOS3
SCHEMBL30868505 0.75 HTT (0.46) CSNK1A1CLK4PIK3CAPIK3CDNOS3
SCHEMBL338485 0.75 HTT (0.46) CSNK1A1CLK4PIK3CAPIK3CDNOS3
SCHEMBL1457800 0.74 CSNK1A1 (0.44) CSNK1A1CLK4PIK3CAPIK3CDNOS3
SCHEMBL30971228 0.74 CSNK1A1 (0.44) CSNK1A1CLK4PIK3CAPIK3CDNOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed