SCHEMBL20157979

SCHEMBL20157979

CCS(=O)(=O)Nc1cc(Br)c(C(=O)c2ccc(C)cc2)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.43
LMNA P02545 5/20 0.43
HTT P42858 5/20 0.43
TP53 P04637 2/20 0.43
KMT2A Q03164 1/20 0.43
HPGD P15428 4/20 0.42
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 1/20 0.42
CCR9 P51686 2/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
HSD17B10 Q99714 2/20 0.38
POLB P06746 1/20 0.38
CYP1A2 P05177 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
RAB9A P51151 1/20 0.37
MRGPRX1 Q96LB2 1/20 0.37
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157971 0.80 NPC1 (0.44) MAPTLMNAHTTTP53KMT2A
SCHEMBL28469745 0.79 KMT2A (0.47) MAPTKMT2AHPGDALDH1A1KDM4E
SCHEMBL20157980 0.78 LMNA (0.38) MAPTLMNAHTTTP53KMT2A
SCHEMBL20157997 0.77 MAPT (0.40) MAPTLMNAHTTTP53KMT2A
SCHEMBL20157667 0.77 MAPT (0.43) MAPTLMNAHTTTP53KMT2A
SCHEMBL20157705 0.76 MAPT (0.49) MAPTLMNAHTTALDH1A1L3MBTL1
SCHEMBL20157995 0.74 MAPT (0.44) MAPTLMNAHTTALDH1A1CA12
SCHEMBL20157982 0.74 LCK (0.39) MAPTLMNAHTTTP53HPGD
SCHEMBL20157492 0.73 MAPT (0.57) MAPTLMNAHTTHPGDALDH1A1
SCHEMBL21362817 0.72 HPGD (0.39) MAPTLMNAHPGDALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed