SCHEMBL21362817

SCHEMBL21362817

C=Cc1ccc(C(=O)c2cc(F)c(NS(=O)(=O)CC)cc2Br)cc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.39
ALDH1A1 P00352 3/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
PSIP1 O75475 1/20 0.37
LMNA P02545 2/20 0.37
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
MCL1 Q07820 2/20 0.35
PGR P06401 1/20 0.34
MRGPRX1 Q96LB2 3/20 0.33
NR2F2 P24468 1/20 0.33
BRAF P15056 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157667 0.87 MAPT (0.43) HPGDALDH1A1MAPTKDM4EPSIP1
SCHEMBL20157971 0.85 NPC1 (0.44) HPGDALDH1A1MAPTKDM4EPSIP1
SCHEMBL21362630 0.77 HPGD (0.38) HPGDALDH1A1MAPTKDM4ELMNA
SCHEMBL20157477 0.75 ALDH1A1 (0.52) ALDH1A1MAPTKDM4ELMNA
SCHEMBL21550169 0.74 KMT2A (0.44) HPGDALDH1A1MAPTKDM4EPSIP1
SCHEMBL20157979 0.72 MAPT (0.43) HPGDALDH1A1MAPTKDM4ELMNA
SCHEMBL20157891 0.72 KDM1A (0.43) HPGDALDH1A1MAPTLMNA
SCHEMBL21362746 0.70 TAS1R3 (0.35) HPGDMAPTTAS1R3TAS1R1MCL1
SCHEMBL20158009 0.68 GAA (0.38) ALDH1A1MAPTKDM4ELMNA
SCHEMBL16658378 0.68 PSIP1 (0.49) HPGDALDH1A1MAPTKDM4EPSIP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed