SCHEMBL20158832

SCHEMBL20158832

COc1ccc(C(=O)n2c3ccc(Br)cc3c3c(C)nn(C)c32)cc1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.49
ELANE P08246 4/20 0.45
ALDH1A1 P00352 2/20 0.45
MCL1 Q07820 1/20 0.45
AKR1C3 P42330 4/20 0.44
AKR1C2 P52895 3/20 0.44
PTGS2 P35354 3/20 0.42
PIK3R1 P27986 1/20 0.41
PIK3CA P42336 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20139087 0.89 ELANE (0.53) MAPK8ELANEALDH1A1MCL1AKR1C3
SCHEMBL24200445 0.87 MAPK8 (0.53) MAPK8ELANEALDH1A1PTGS2
SCHEMBL20159077 0.85 LMNA (0.55) ELANEAKR1C3AKR1C2PTGS2
SCHEMBL20138831 0.79 CNR1 (0.43) ELANEALDH1A1
SCHEMBL24200422 0.78 MAPK8 (0.51) MAPK8ELANEALDH1A1
SCHEMBL20138825 0.76 ELANE (0.54) MAPK8ELANE
SCHEMBL20158841 0.74 ELANE (0.56) ELANEAKR1C3AKR1C2PTGS2
SCHEMBL20147125 0.72 P2RX4 (0.50) ELANEALDH1A1PTGS2
SCHEMBL20158843 0.69 ELANE (0.43) ELANEALDH1A1MCL1
SCHEMBL20158839 0.67 ELANE (0.42) MAPK8ELANEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018087389-A1 SELECTIVE INHIBITORS OF GENOTOXIC STRESS-INDUCED IKK/NF-kB PATHWAYS MAX-DELBRÜCK-CENTRUM FÜR MOLEKULARE MEDIZIN IN DER HELMHOLTZ-GEMEINSCHAFT (DE) 2018-05-17 WO disclosed