SCHEMBL24200422

SCHEMBL24200422

Cc1nn(C)c2c1c1cc(Br)ccc1n2C(=O)c1ccccc1Br

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 2/20 0.51
ELANE P08246 5/20 0.40
CNR2 P34972 1/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPK9 P45984 1/20 0.36
POLB P06746 1/20 0.36
PRNP P04156 1/20 0.35
PPARG P37231 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
NR2E3 Q9Y5X4 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
CA12 O43570 1/20 0.34
CA9 Q16790 1/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158839 0.89 ELANE (0.42) MAPK8ELANECNR2ALDH1A1PRNP
SCHEMBL20138831 0.87 CNR1 (0.43) ELANECNR2ALDH1A1POLB
SCHEMBL24200445 0.86 MAPK8 (0.53) MAPK8ELANEALDH1A1POLBPRNP
SCHEMBL20158832 0.78 MAPK8 (0.49) MAPK8ELANEALDH1A1
SCHEMBL20158843 0.77 ELANE (0.43) ELANECNR2ALDH1A1
SCHEMBL20138825 0.75 ELANE (0.54) MAPK8ELANEPRNPPPARGRXFP1
SCHEMBL20159077 0.71 LMNA (0.55) ELANEPPARG
SCHEMBL20147125 0.71 P2RX4 (0.50) ELANEALDH1A1
SCHEMBL20139087 0.67 ELANE (0.53) MAPK8ELANEALDH1A1
SCHEMBL7059986 0.67 CNR2 (0.39) ELANECNR2ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538529-B1 SELECTIVE INHIBITORS OF GENOTOXIC STRESS-INDUCED IKK/NF-KB PATHWAYS MAX DELBRUECK CENTRUM FUER MOLEKULARE MEDIZIN HELMHOLTZ GEMEINSCHAFT (DE) 2022-01-19 EP disclosed