SCHEMBL20159004

SCHEMBL20159004

N#Cc1c(F)cccc1P

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
KDM4E B2RXH2 4/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TRPV4 Q9HBA0 2/20 0.41
CUL4A Q13619 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TAS1R2 Q8TE23 1/20 0.35
MAPT P10636 2/20 0.34
DRD2 P14416 1/20 0.34
HTR2A P28223 1/20 0.34
HRH1 P35367 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ADORA1 P30542 2/20 0.33
ADORA2A P29274 1/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
CACNA1B Q00975 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL186269 0.83 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDHSD17B10TRPV4
Cyanide SCHEMBL28871133 0.78 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDHSD17B10TRPV4
SCHEMBL19062287 0.76 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHSD17B10TRPV4
SCHEMBL186554 0.74 KDM4E (0.44) ALDH1A1KDM4EHPGDHSD17B10TRPV4
SCHEMBL186023 0.73 KDM4E (0.47) ALDH1A1KDM4EHPGDHSD17B10TAS1R3
SCHEMBL421862 0.73 ALDH1A1 (0.43) ALDH1A1KDM4EHPGDHSD17B10TRPV4
SCHEMBL286715 0.73 CYP1A2 (0.50) ALDH1A1KDM4EHPGDHSD17B10TRPV4
SCHEMBL3154084 0.73 ALDH1A1 (0.43) ALDH1A1KDM4EHPGDHSD17B10TRPV4
SCHEMBL525892 0.73 ALDH1A1 (0.43) ALDH1A1KDM4EHPGDHSD17B10TRPV4
SCHEMBL29555331 0.73 KDM4E (0.43) ALDH1A1KDM4EHPGDHSD17B10TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed