SCHEMBL20159100

SCHEMBL20159100

NN1CCc2ccncc2CC1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.59
CHRNB2 P17787 1/20 0.53
CHRNA4 P43681 1/20 0.53
EED O75530 1/20 0.38
HPGD P15428 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
GAA P10253 1/20 0.33
NAMPT P43490 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18630000 0.88 SIGMAR1 (0.50) SIGMAR1CHRNB2CHRNA4EEDHPGD
SCHEMBL15025467 0.88 SIGMAR1 (0.50) SIGMAR1CHRNB2CHRNA4EEDHPGD
SCHEMBL20159085 0.81 SIGMAR1 (0.61) SIGMAR1CHRNB2CHRNA4
SCHEMBL8348679 0.79
SCHEMBL9965975 0.76 MAOA (0.59) SIGMAR1CHRNB2CHRNA4EED
5,6,7,8-Tetrahydroisoquinoline SCHEMBL28211 0.75 SIGMAR1 (1.00) SIGMAR1CHRNB2CHRNA4
SCHEMBL29518090 0.75
SCHEMBL2388666 0.75
SCHEMBL14730735 0.74 SIGMAR1 (0.46) SIGMAR1CHRNB2CHRNA4NAMPT
SCHEMBL9965909 0.73 MAOA (0.55) SIGMAR1CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed