SCHEMBL20159207

SCHEMBL20159207

CC1(C)CC(c2ccc(N)cc2)=NN(CCN2C(=O)c3ccccc3C2=O)C1=O

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTR1A P08908 2/20 0.38
LMNA P02545 2/20 0.38
ACHE P22303 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GLS O94925 1/20 0.34
NPC1 O15118 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159747 0.89 GSK3B (0.40) MEN1GAAKMT2ACYP1A2CYP2C9
SCHEMBL20138842 0.81 PDE4B (0.40) MEN1GAAKMT2ALMNASMN1; SMN2
SCHEMBL20159539 0.79 HRH3 (0.36) CYP1A2CYP2C19
SCHEMBL20138839 0.79 CYP19A1 (0.39) MEN1KMT2ALMNASMN1; SMN2NPC1
SCHEMBL20159716 0.79 PDE4B (0.36) MEN1KMT2ALMNASMN1; SMN2NPC1
SCHEMBL20159528 0.77 PDE4B (0.40) MEN1KMT2ACYP2C9
SCHEMBL20159426 0.76 CYP19A1 (0.38) MEN1KMT2A
SCHEMBL20159516 0.75 PDE4B (0.34) MEN1KMT2A
SCHEMBL20159396 0.75 HRH3 (0.36) MEN1KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL20142920 0.75 CYP19A1 (0.45) MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021013693-A1 ANTIBODY DRUG CONJUGATES (ADCS) WITH NAMPT INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2021-01-28 WO disclosed
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed