SCHEMBL20159528

SCHEMBL20159528

COCCCN1N=C(c2ccc(N)cc2)CC(C)(C)C1=O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 4/20 0.40
REN P00797 9/20 0.36
CYP2D6 P10635 5/20 0.35
CYP2C9 P11712 5/20 0.35
KCNH2 Q12809 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CYP19A1 P11511 1/20 0.34
CYP3A4 P08684 4/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159716 0.93 PDE4B (0.36) PDE4BKCNH2HRH3CYP19A1MEN1
SCHEMBL20159532 0.88 SMN1; SMN2 (0.41) PDE4BRENCYP2D6CYP2C9KCNH2
SCHEMBL20138842 0.83 PDE4B (0.40) PDE4BCYP19A1MEN1KMT2AALDH1A1
SCHEMBL20138839 0.81 CYP19A1 (0.39) PDE4BCYP19A1MEN1KMT2AALDH1A1
SCHEMBL20138895 0.81 SMN1; SMN2 (0.43) PDE4BKCNH2HRH3MEN1KMT2A
SCHEMBL20142970 0.80 TP53 (0.36) PDE4BMEN1KMT2A
SCHEMBL20159539 0.79 HRH3 (0.36) CYP2D6HRH3CYP19A1ALDH1A1
SCHEMBL20159426 0.78 CYP19A1 (0.38) PDE4BKCNH2HRH3CYP19A1MEN1
SCHEMBL20159396 0.77 HRH3 (0.36) PDE4BCYP2C9HRH3CYP19A1MEN1
SCHEMBL20159516 0.77 PDE4B (0.34) PDE4BCYP19A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed