SCHEMBL20142920

SCHEMBL20142920

CN1N=C(c2ccc(N)cc2)CC(C)(C)C1=O

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 11/20 0.45
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KEAP1 Q14145 1/20 0.34
BACE1 P56817 2/20 0.33
REN P00797 1/20 0.33
APP P05067 1/20 0.33
BACE2 Q9Y5Z0 1/20 0.33
MAPT P10636 1/20 0.33
RECQL P46063 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20142960 0.84 SMN1; SMN2 (0.41) MEN1KMT2AL3MBTL1KDM4EALDH1A1
SCHEMBL20138839 0.81 CYP19A1 (0.39) CYP19A1MEN1KMT2AL3MBTL1KDM4E
SCHEMBL20138842 0.80 PDE4B (0.40) CYP19A1MEN1KMT2AL3MBTL1KDM4E
SCHEMBL20142933 0.80 PDE4B (0.45) CYP19A1MEN1KMT2AL3MBTL1KDM4E
SCHEMBL20159211 0.79 SMN1; SMN2 (0.40) MEN1KMT2AL3MBTL1KDM4EALDH1A1
SCHEMBL20159716 0.78 PDE4B (0.36) CYP19A1MEN1KMT2AL3MBTL1ALDH1A1
SCHEMBL20159426 0.77 CYP19A1 (0.38) CYP19A1MEN1KMT2AL3MBTL1
SCHEMBL20159203 0.77 PDE4D (0.44) CYP19A1MEN1KMT2AL3MBTL1KDM4E
SCHEMBL20159509 0.77 PDE4B (0.46) CYP19A1SMN1; SMN2
SCHEMBL20159396 0.76 HRH3 (0.36) CYP19A1MEN1KMT2AL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed