SCHEMBL20159462

SCHEMBL20159462

CN1N=C(c2ccc(NC(=O)N3CCc4cccnc43)cc2)CC(C)(C)C1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 6/20 0.41
NPC1 O15118 5/20 0.41
RAB9A P51151 5/20 0.41
SMN1; SMN2 Q16637 5/20 0.41
NFKB1 P19838 3/20 0.41
NFKB2 Q00653 3/20 0.41
RELA Q04206 3/20 0.41
CRBN Q96SW2 2/20 0.39
MTNR1A P48039 1/20 0.39
ROCK2 O75116 2/20 0.38
ROCK1 Q13464 2/20 0.38
HTR2C P28335 3/20 0.38
HTR2B P41595 1/20 0.38
PKM P14618 2/20 0.38
MAPT P10636 1/20 0.38
MAOB P27338 1/20 0.38
FGFR4 P22455 1/20 0.37
POLB P06746 1/20 0.37
HTR2A P28223 1/20 0.37
CACNA1H O95180 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159221 0.84 NAMPT (0.47) ROCK2
SCHEMBL20159441 0.75 NAMPT (0.52)
SCHEMBL20159469 0.75 NAMPT (0.52)
SCHEMBL20159409 0.72 NAMPT (0.53) ROCK2
SCHEMBL20138871 0.70 NAMPT (0.52) ROCK2
SCHEMBL20159518 0.70 NAMPT (0.53) ROCK2
SCHEMBL20139005 0.69 NAMPT (0.57) ROCK2
SCHEMBL20159251 0.69 NAMPT (0.39) ROCK2
SCHEMBL20159429 0.65 ROCK2 (0.56) ROCK2
SCHEMBL20142920 0.65 CYP19A1 (0.45) SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed