SCHEMBL20159532

SCHEMBL20159532

COCCCN1N=C(c2ccc(Br)cc2)CC(C)(C)C1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
PDE4B Q07343 5/20 0.40
KCNH2 Q12809 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
PAX8 Q06710 1/20 0.34
ALDH1A1 P00352 3/20 0.33
REN P00797 3/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
GAA P10253 1/20 0.33
FPR1 P21462 1/20 0.33
HTT P42858 1/20 0.33
HIF1A Q16665 1/20 0.33
MAPT P10636 2/20 0.33
LMNA P02545 1/20 0.32
ITGB2 P05107 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20138895 0.93 SMN1; SMN2 (0.43) SMN1; SMN2NPC1RAB9APDE4BKCNH2
SCHEMBL20159528 0.88 PDE4B (0.40) PDE4BKCNH2HRH3KMT2AMEN1
SCHEMBL20142913 0.81 SMN1; SMN2 (0.39) SMN1; SMN2NPC1RAB9APDE4BKMT2A
SCHEMBL20159716 0.81 PDE4B (0.36) SMN1; SMN2NPC1RAB9APDE4BKCNH2
SCHEMBL20159737 0.79 RAB9A (0.36) SMN1; SMN2NPC1RAB9AHRH3ALDH1A1
SCHEMBL20138970 0.78 FPR1 (0.37) SMN1; SMN2NPC1RAB9APDE4BKMT2A
SCHEMBL20159747 0.77 GSK3B (0.40) SMN1; SMN2RAB9AKMT2AMEN1ALDH1A1
SCHEMBL20159360 0.77 NPC1 (0.44) SMN1; SMN2NPC1RAB9APDE4BHRH3
SCHEMBL20159374 0.77 SMN1; SMN2 (0.39) SMN1; SMN2NPC1RAB9APDE4BKMT2A
SCHEMBL20142960 0.76 SMN1; SMN2 (0.41) SMN1; SMN2NPC1RAB9APDE4BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed