SCHEMBL20159904

SCHEMBL20159904

Nc1ccc(Oc2ccc(F)cc2F)c(-c2ccc3nncn3c2)c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.41
BRD4 O60885 7/20 0.41
MLLT1 Q03111 1/20 0.41
SCN5A Q14524 1/20 0.39
TGFBR1 P36897 1/20 0.38
PIK3CA P42336 1/20 0.38
DNMT1 P26358 1/20 0.36
ADORA2A P29274 2/20 0.35
ADORA2B P29275 2/20 0.35
ADORA1 P30542 2/20 0.35
SCN4A P35499 1/20 0.34
BRD2 P25440 1/20 0.33
BRD3 Q15059 1/20 0.33
BRDT Q58F21 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20160241 0.79 PIM1 (0.44) MAPK14BRD4
SCHEMBL20160416 0.78 BRD4 (0.55) BRD4ADORA2BBRD2BRD3BRDT
SCHEMBL20160293 0.78 BRD4 (0.43) MAPK14BRD4SCN4A
SCHEMBL15549928 0.74 BRD4 (0.53) BRD4BRD2BRD3BRDT
SCHEMBL29548595 0.71 BRD4 (0.47) MAPK14BRD4ADORA2A
SCHEMBL20160236 0.70 BRD4 (0.43) MAPK14BRD4ADORA2ABRD2BRD3
SCHEMBL20159919 0.70 BRD4 (0.47) MAPK14BRD4
SCHEMBL21904846 0.70 BRD4 (0.64) BRD4BRD2BRD3BRDT
SCHEMBL20159911 0.70 BRD4 (0.43) MAPK14BRD4BRD2BRD3
SCHEMBL15553259 0.69 BRD4 (0.71) BRD4BRD2BRD3BRDT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed