SCHEMBL20160282

SCHEMBL20160282

CCNc1ccc(Oc2ccc(F)cc2F)c(-c2cccc3c2C(=O)NC3=O)c1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 20/20 0.49
BRD2 P25440 1/20 0.42
ADORA2B P29275 1/20 0.42
TSPO P30536 1/20 0.42
EP300 Q09472 1/20 0.42
BRD3 Q15059 1/20 0.42
BRDT Q58F21 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159920 0.80 BRD4 (0.48) BRD4BRD2BRD3BRDT
SCHEMBL20160047 0.69 BRD4 (0.59) BRD4BRD2ADORA2BTSPOEP300
SCHEMBL6341593 0.67 KDM4E (0.58)
SCHEMBL16765616 0.66 BRD4 (1.00) BRD4
SCHEMBL15552165 0.65 BRD4 (0.78) BRD4
SCHEMBL262473 0.65 GSK3B (0.50)
SCHEMBL22032796 0.65 NTRK1 (0.46)
SCHEMBL21904838 0.65 BRD4 (0.64) BRD4BRD2ADORA2BTSPOEP300
SCHEMBL20160417 0.65 BRD4 (0.42) BRD4
SCHEMBL16654653 0.65 BRD4 (0.63) BRD4BRD2ADORA2BTSPOEP300

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed