SCHEMBL20159971

SCHEMBL20159971

Cc1ccc(Oc2nc(I)nn2C(C)C)cc1C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AR P10275 9/20 0.33
CDK8 P49336 1/20 0.33
RHEB Q15382 1/20 0.33
ESR1 P03372 1/20 0.33
MGLL Q99685 1/20 0.32
PSEN1 P49768 2/20 0.32
PSEN2 P49810 2/20 0.32
APH1B Q8WW43 2/20 0.32
NCSTN Q92542 2/20 0.32
APH1A Q96BI3 2/20 0.32
PSENEN Q9NZ42 2/20 0.32
ABL1 P00519 1/20 0.31
SRC P12931 1/20 0.31
P2RX3 P56373 1/20 0.31
CYP1A2 P05177 1/20 0.31
KDR P35968 1/20 0.31
S1PR1 P21453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20142944 0.85 AR (0.33) ARCDK8RHEBESR1MGLL
SCHEMBL23504842 0.81 LMNA (0.39) CDK8PSEN1PSEN2APH1BNCSTN
SCHEMBL23504812 0.78 CDK1 (0.35)
SCHEMBL23504771 0.78 HTR2A (0.41)
SCHEMBL20159299 0.73 HTR2A (0.37) ARCDK8MGLLABL1SRC
SCHEMBL20159274 0.73 HTR2A (0.37) ARMGLLPSEN1PSEN2APH1B
SCHEMBL20159329 0.72 PLA2G7 (0.40)
SCHEMBL29623386 0.72 PLA2G7 (0.40)
SCHEMBL20138679 0.71 AR (0.32) ARMGLLS1PR1
SCHEMBL20159726 0.71 KCNH2 (0.39) ARCDK8MGLLKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018087018-A1 PHENOXYTRIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2018-05-17 WO disclosed