SCHEMBL20160417

SCHEMBL20160417

CCNc1ccc(Oc2ccc(F)cc2F)c(-c2ccc3nncn3n2)c1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 16/20 0.42
NPC1 O15118 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20160293 0.81 BRD4 (0.43) BRD4NPC1HTTSMN1; SMN2KDM4E
SCHEMBL20159984 0.71 SMN1; SMN2 (0.35) BRD4NPC1HTTSMN1; SMN2KDM4E
SCHEMBL20160273 0.70 SMN1; SMN2 (0.56) BRD4SMN1; SMN2KDM4E
SCHEMBL20159838 0.69 BRD4 (0.56) BRD4
SCHEMBL20160416 0.68 BRD4 (0.55) BRD4
SCHEMBL20159922 0.67 BRD4 (0.47) BRD4
SCHEMBL20160303 0.65 BRD4 (0.58) BRD4
SCHEMBL20160282 0.65 BRD4 (0.49) BRD4
SCHEMBL20159910 0.65 NPC1 (0.39) BRD4NPC1MAPT
SCHEMBL20160024 0.64 BRD4 (0.45) BRD4SMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed