SCHEMBL20160415

SCHEMBL20160415

CCOC(=O)Nc1cc(Cl)nn2cnnc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
BRPF1 P55201 2/20 0.40
HPGD P15428 2/20 0.40
TRIM24 O15164 1/20 0.39
BRD4 O60885 1/20 0.39
BRD1 O95696 1/20 0.39
TAF1 P21675 1/20 0.39
BRD2 P25440 1/20 0.39
SMARCA4 P51532 1/20 0.39
BPTF Q12830 1/20 0.39
BRDT Q58F21 1/20 0.39
ATAD2 Q6PL18 1/20 0.39
PBRM1 Q86U86 1/20 0.39
TAF1L Q8IZX4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20160359 0.86 CYP2C9 (0.43) ALDH1A1CYP1A2CYP2C9CYP2C19SMN1; SMN2
SCHEMBL140145 0.84 KDM4E (0.39) ALDH1A1CYP1A2CYP2C9SMN1; SMN2KMT2A
SCHEMBL105064 0.82 BRD9 (0.45) BRD4BRD2CREBBPBRD9TNKS
SCHEMBL105123 0.79 BAZ2B (0.41) ALDH1A1CYP1A2CYP2C9SMN1; SMN2KMT2A
SCHEMBL20160220 0.78 BRPF1 (0.58) ALDH1A1CYP1A2CYP2C9CYP2C19SMN1; SMN2
SCHEMBL5057070 0.71 KMT2A (0.41) ALDH1A1CYP1A2CYP2C9SMN1; SMN2KMT2A
SCHEMBL21354900 0.68 BRD9 (0.39) ALDH1A1KMT2ABRD4BRD9KDM4E
SCHEMBL104901 0.67 KDM4E (0.40) ALDH1A1CYP1A2CYP2C9SMN1; SMN2KMT2A
SCHEMBL20160351 0.67 BRPF1 (0.57) ALDH1A1CYP1A2CYP2C9CYP2C19SMN1; SMN2
SCHEMBL3784358 0.67 ALDH1A1 (0.73) ALDH1A1CYP1A2CYP2C9CYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed