Iodide

Iodide

SCHEMBL2016181

CCn1c(COC(=O)c2nc(Cl)c(N)nc2N)[n+](C)c2cc(-c3ccc(OC)cc3)ccc21.[I-]

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCNN1A P37088 5/20 0.38
MAPT P10636 2/20 0.36
NPC1 O15118 1/20 0.36
NLRP3 Q96P20 1/20 0.36
GABRA2 P47869 2/20 0.36
GABRB2 P47870 2/20 0.36
MEN1 O00255 1/20 0.35
APAF1 O14727 1/20 0.35
USP2 O75604 1/20 0.35
HSP90AA1 P07900 1/20 0.35
NTSR1 P30989 1/20 0.35
UBE2N P61088 1/20 0.35
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 2/20 0.35
PPARG P37231 1/20 0.34
TARBP2 Q15633 2/20 0.34
PDCD4 Q53EL6 1/20 0.34
DHODH Q02127 1/20 0.34
PDE5A O76074 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12635760 0.99 SCNN1A (0.38) SCNN1AMAPTNPC1NLRP3GABRA2
Iodide SCHEMBL2018286 0.95 SCNN1A (0.38) SCNN1AMAPTNPC1NLRP3GABRA2
SCHEMBL12636304 0.94 SCNN1A (0.38) SCNN1AMAPTNPC1NLRP3GABRA2
Iodide SCHEMBL2053822 0.88 SCNN1A (0.36) SCNN1AMAPTNPC1NLRP3SMN1; SMN2
Iodide SCHEMBL2013734 0.87 SCNN1A (0.41) SCNN1AMAPTALDH1A1SMN1; SMN2
Iodide SCHEMBL2014693 0.87 SCNN1A (0.37) SCNN1AMAPTNPC1NLRP3GABRA2
SCHEMBL12635745 0.86 SCNN1A (0.42) SCNN1AMAPTALDH1A1SMN1; SMN2
Iodide SCHEMBL2016509 0.86 SCNN1A (0.39) SCNN1AMAPTGABRA2GABRB2MEN1
Iodide SCHEMBL2017093 0.86 ELANE (0.33) GABRA2GABRB2MEN1APAF1USP2
SCHEMBL12636287 0.85 SCNN1A (0.39) SCNN1AMAPTGABRA2GABRB2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO claimed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed