Iodide

Iodide

SCHEMBL2016509

COc1ccc(-c2ccc3c(c2)n(C)c(COC(=O)c2nc(Cl)c(N)nc2N)[n+]3C)cc1.[I-]

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCNN1A P37088 5/20 0.39
GABRA2 P47869 2/20 0.37
GABRB2 P47870 2/20 0.37
PARP1 P09874 1/20 0.35
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
DHODH Q02127 1/20 0.33
TARBP2 Q15633 1/20 0.33
PDCD4 Q53EL6 1/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
THRB P10828 1/20 0.33
PTPN11 Q06124 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12636287 0.99 SCNN1A (0.39) SCNN1AGABRA2GABRB2PARP1ALDH1A1
Iodide SCHEMBL2016658 0.94 SCNN1A (0.38) SCNN1AGABRA2GABRB2ALDH1A1LMNA
Iodide SCHEMBL2018286 0.90 SCNN1A (0.38) SCNN1AGABRA2GABRB2ALDH1A1MEN1
SCHEMBL12636304 0.89 SCNN1A (0.38) SCNN1AGABRA2GABRB2ALDH1A1MEN1
Iodide SCHEMBL2021198 0.87 MAPT (0.36) GABRA2GABRB2ALDH1A1LMNAMAPT
Iodide SCHEMBL2017463 0.86 KDM4E (0.33) SCNN1AGABRA2GABRB2ALDH1A1LMNA
Iodide SCHEMBL2016181 0.86 SCNN1A (0.38) SCNN1AGABRA2GABRB2ALDH1A1MEN1
SCHEMBL12635733 0.86 MAPT (0.36) GABRA2GABRB2ALDH1A1LMNAMAPT
Iodide SCHEMBL2016304 0.85 GABRA2 (0.32) SCNN1AGABRA2GABRB2LMNAKMT2A
SCHEMBL12635760 0.85 SCNN1A (0.38) SCNN1AGABRA2GABRB2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO claimed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed