SCHEMBL2016501

SCHEMBL2016501

OCC1CCCN(c2c(CCNc3ncnc4[nH]cnc34)cc(Cl)c3cccnc23)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KHK P50053 1/20 0.36
METAP2 P50579 3/20 0.35
MAP4K4 O95819 2/20 0.35
KDM4E B2RXH2 3/20 0.33
LMNA P02545 3/20 0.33
MAPT P10636 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
TDP1 Q9NUW8 3/20 0.33
HTT P42858 3/20 0.33
ALDH1A1 P00352 1/20 0.33
MPI P34949 1/20 0.33
ATR Q13535 1/20 0.33
ATRIP Q8WXE1 1/20 0.33
CCR4 P51679 1/20 0.32
KMT2A Q03164 3/20 0.32
RAB9A P51151 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
USP2 O75604 1/20 0.32
MAPK1 P28482 1/20 0.32
NOD2 Q9HC29 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL2013265 0.94 KHK (0.33) KHKMETAP2MAP4K4BTK
SCHEMBL2016811 0.89 METAP2 (0.34) METAP2KDM4ELMNAMAPTSMN1; SMN2
SCHEMBL2014977 0.88 SLC40A1 (0.38) METAP2KDM4ELMNAMAPTSMN1; SMN2
SCHEMBL2014980 0.88 SLC40A1 (0.38) METAP2KDM4ELMNAMAPTSMN1; SMN2
SCHEMBL2017050 0.86 SLC40A1 (0.40) METAP2KDM4ELMNAMAPTSMN1; SMN2
SCHEMBL2015211 0.84 AXL (0.32) METAP2KDM4ELMNAMAPTSMN1; SMN2
SCHEMBL2016495 0.83 PIK3CD (0.42) KHKMAP4K4KDM4ELMNAMAPT
SCHEMBL2016578 0.83 CNR2 (0.38) RAB9AL3MBTL1BTKNPC1
SCHEMBL2012932 0.82 ABCC1 (0.33) METAP2KDM4ELMNAMAPTSMN1; SMN2
SCHEMBL2013366 0.82 CCR4 (0.37) METAP2LMNAMAPTSMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO claimed