SCHEMBL2016536

SCHEMBL2016536

CCOc1ccc2nc(CNC(=O)c3nc(Cl)c(N)nc3N)n(CC)c2c1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.42
ACSS2 Q9NR19 5/20 0.41
ACACB O00763 1/20 0.41
MTNR1A P48039 4/20 0.39
MTNR1B P49286 4/20 0.39
SCNN1A P37088 3/20 0.39
KDM4E B2RXH2 1/20 0.38
USP2 O75604 1/20 0.38
POLB P06746 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
CTSA P10619 1/20 0.38
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2018430 0.93 ACSS2 (0.42) HTTACSS2SCNN1AKCNH2
SCHEMBL2022069 0.92 ACSS2 (0.47) HTTACSS2SCNN1ACTSAKCNH2
SCHEMBL2018438 0.92 SCNN1A (0.44) HTTACSS2MTNR1AMTNR1BSCNN1A
SCHEMBL12635701 0.91 ACSS2 (0.49) HTTACSS2MTNR1AMTNR1BSCNN1A
SCHEMBL12635952 0.90 HTT (0.41) HTTACSS2MTNR1AMTNR1BSCNN1A
SCHEMBL2015793 0.90 KCNH2 (0.49) HTTACSS2SCNN1AKDM4EKCNH2
SCHEMBL16882065 0.89 SCNN1A (0.40) HTTACSS2SCNN1AKCNH2
SCHEMBL2017976 0.88 HTT (0.40) HTTACSS2SCNN1ACTSAKCNH2
SCHEMBL21335806 0.88 SCNN1A (0.39) HTTACSS2SCNN1AKCNH2
SCHEMBL2040435 0.88 HTT (0.45) HTTACSS2CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed