SCHEMBL2040435

SCHEMBL2040435

CCn1c(CNC(=O)c2nc(Cl)c(N)nc2N)nc2ccc(Cl)cc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.45
ALDH1A1 P00352 1/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ACSS2 Q9NR19 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CTSA P10619 2/20 0.38
ADORA2A P29274 1/20 0.38
TP53 P04637 3/20 0.37
GRM5 P41594 1/20 0.37
NTRK1 P04629 1/20 0.37
NTRK2 Q16620 1/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2016331 0.91 HTT (0.52) HTTALDH1A1GLAGAAMAPT
SCHEMBL2014823 0.91 HTT (0.45) HTTMEN1KMT2ACTSATP53
SCHEMBL2016153 0.90 HTT (0.44) HTTALDH1A1GLAGAAMAPT
SCHEMBL2017836 0.89 HTT (0.46) HTTALDH1A1ACSS2MEN1KMT2A
Iodide SCHEMBL2019625 0.89 HTT (0.43) HTTALDH1A1GLAGAAMAPT
SCHEMBL2020338 0.89 HTT (0.46) HTTALDH1A1GLAGAAMAPT
SCHEMBL2020396 0.89 HTT (0.48) HTTACSS2MEN1KMT2ATP53
SCHEMBL2018438 0.88 SCNN1A (0.44) HTTMAPTSMN1; SMN2ACSS2TP53
SCHEMBL12635756 0.88 HTT (0.49) HTTACSS2MEN1KMT2ATSHR
SCHEMBL2015344 0.88 HTT (0.47) HTTMAPTSMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed