SCHEMBL2015793

SCHEMBL2015793

CCn1c(CNC(=O)c2nc(Cl)c(N)nc2N)nc2ccc(OCc3ccccc3)cc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.49
ACSS2 Q9NR19 7/20 0.48
HTT P42858 1/20 0.42
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
GLA P06280 2/20 0.40
HPGD P15428 2/20 0.40
HSD17B10 Q99714 2/20 0.40
SCNN1A P37088 2/20 0.40
MAPT P10636 2/20 0.40
NPC1 O15118 1/20 0.40
CYP1A2 P05177 1/20 0.40
GAA P10253 1/20 0.40
CYP2D6 P10635 1/20 0.40
NFKB1 P19838 1/20 0.40
THPO P40225 1/20 0.40
HIF1A Q16665 1/20 0.40
FTO Q9C0B1 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
S1PR3 Q99500 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2016536 0.90 HTT (0.42) KCNH2ACSS2HTTKDM4ESCNN1A
SCHEMBL2022069 0.89 ACSS2 (0.47) KCNH2ACSS2HTTSCNN1AMEN1
SCHEMBL2018430 0.88 ACSS2 (0.42) KCNH2ACSS2HTTSCNN1AS1PR3
SCHEMBL2018438 0.87 SCNN1A (0.44) ACSS2HTTSCNN1AMAPT
SCHEMBL12635701 0.86 ACSS2 (0.49) KCNH2ACSS2HTTSCNN1A
SCHEMBL2017976 0.85 HTT (0.40) KCNH2ACSS2HTTSCNN1AMEN1
SCHEMBL12635952 0.85 HTT (0.41) KCNH2ACSS2HTTALDH1A1GLA
SCHEMBL2014823 0.84 HTT (0.45) HTTHSD17B10SCNN1ACYP1A2CYP2D6
SCHEMBL21335806 0.83 SCNN1A (0.39) KCNH2ACSS2HTTSCNN1A
SCHEMBL2040435 0.83 HTT (0.45) ACSS2HTTALDH1A1GLAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed