SCHEMBL20169647

SCHEMBL20169647

BOC(=O)c1nc(C)c(C)nc1N

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.37
HPGD P15428 3/20 0.37
GAA P10253 1/20 0.37
CYP1A2 P05177 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
KDM4E B2RXH2 5/20 0.34
HSD17B10 Q99714 2/20 0.34
LMNA P02545 4/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PKM P14618 1/20 0.33
HTT P42858 1/20 0.33
RECQL P46063 1/20 0.33
PDPK1 O15530 1/20 0.32
MAPT P10636 1/20 0.31
TP53 P04637 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16418573 0.81 NPSR1 (0.56) ALDH1A1HPGDGAACYP1A2CA12
SCHEMBL29977899 0.81 NPSR1 (0.56) ALDH1A1HPGDGAACYP1A2CA12
SCHEMBL3800959 0.76 GABRP (0.41) ALDH1A1HPGDCA12CA2CA9
SCHEMBL26039163 0.76 PDPK1 (0.50) ALDH1A1HPGDGAACYP1A2KDM4E
SCHEMBL30793018 0.76 PDPK1 (0.50) ALDH1A1HPGDGAACYP1A2KDM4E
SCHEMBL31093865 0.73 HCRTR1 (0.34) ALDH1A1HPGDGAA
Lithium Ion SCHEMBL17781253 0.72 ALDH1A1 (0.34) ALDH1A1HPGDGAACYP1A2CA12
SCHEMBL13144986 0.71 NPSR1 (0.54) ALDH1A1HPGDGAACYP1A2KDM4E
SCHEMBL20169653 0.69 KDM4E (0.30) ALDH1A1HPGDGAAKDM4EHSD17B10
SCHEMBL6617911 0.67 NPSR1 (0.48) ALDH1A1HPGDGAAKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9975910-B2 Hetero-fused cyclic compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2018-05-22 US disclosed