SCHEMBL20170495

SCHEMBL20170495

Fc1ccc(CCn2cncc2-c2ccccc2C2CCCN2Sc2cnc(N3CCN4CCCC4C3)s2)cc1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.33
HRH3 Q9Y5N1 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
IDO1 P14902 1/20 0.30
CYP2B6 P20813 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20170406 0.84 CYP11B2 (0.33) CYP11B2CYP3A4CYP2D6IDO1CYP2B6
SCHEMBL20169605 0.84 CYP11B2 (0.33) CYP11B2CYP3A4CYP2D6IDO1CYP2B6
SCHEMBL20170435 0.76 ATR (0.31) HRH3
SCHEMBL16720946 0.76 CYP11B2 (0.32) CYP11B2CYP3A4CYP2D6IDO1CYP2B6
SCHEMBL20170514 0.75 KCNH2 (0.32) HRH3
SCHEMBL16730886 0.74 CYP11B2 (0.46) CYP11B2CYP3A4CYP2D6IDO1CYP2B6
SCHEMBL18128805 0.74 CYP11B2 (0.46) CYP11B2CYP3A4CYP2D6IDO1CYP2B6
SCHEMBL20170492 0.74 DRD3 (0.39) CYP11B2HRH3CYP3A4CYP2D6IDO1
SCHEMBL20170477 0.73 SCN9A (0.31)
SCHEMBL20170510 0.71 CYP11B2 (0.42) CYP11B2CYP3A4CYP2D6IDO1CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068391-B1 ARYL LINKED IMIDAZOLE AND TRIAZOLE DERIVATIVES AND METHODS OF USE THEREOF FOR IMPROVING THE PHARMACOKINETICS OF A DRUG MERCK SHARP & DOHME (US) 2018-05-23 EP disclosed