SCHEMBL20170704

SCHEMBL20170704

COC1=CC2CCc3ccc(OC)c(O)c3CC2CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 6/20 0.38
DRD2 P14416 5/20 0.38
F3 P13726 1/20 0.38
CHRM2 P08172 2/20 0.37
CHRM1 P11229 2/20 0.37
CHRM3 P20309 2/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CASP1 P29466 1/20 0.37
CYP2C19 P33261 1/20 0.37
APAF1 O14727 1/20 0.37
BCHE P06276 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
DRD3 P35462 2/20 0.36
DRD4 P21917 1/20 0.36
MTNR1A P48039 2/20 0.36
MTNR1B P49286 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16772366 0.68 DRD1 (0.48) DRD1DRD2F3KDM4ELMNA
SCHEMBL2742544 0.66 DRD1 (0.60) DRD1DRD2F3KDM4ELMNA
SCHEMBL6959755 0.66 CETP (0.44) DRD1DRD2F3KDM4ELMNA
SCHEMBL4128903 0.66 CETP (0.48) DRD1DRD2F3KDM4ELMNA
SCHEMBL16774958 0.65 DRD1 (0.46) DRD1DRD2F3KDM4ELMNA
SCHEMBL20170653 0.63 GAA (0.42) KDM4ECYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL20170665 0.62 CYP3A4 (0.41) DRD1DRD2F3KDM4ECYP1A2
SCHEMBL7363210 0.62 CYP1A2 (0.59) DRD1DRD2F3KDM4ELMNA
SCHEMBL2463383 0.61 ADRA1A (0.47) DRD1DRD2F3KDM4ELMNA
SCHEMBL16210119 0.61 PNMT (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed