SCHEMBL20170653

SCHEMBL20170653

COc1ccc2c(c1O)C1CC(=O)CCC1CC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.42
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
CYP3A4 P08684 3/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 2/20 0.38
HSD17B10 Q99714 2/20 0.38
CYP2C19 P33261 1/20 0.38
HIF1A Q16665 1/20 0.38
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 3/20 0.37
MAPT P10636 2/20 0.37
GLA P06280 1/20 0.37
HPGD P15428 1/20 0.37
RAD52 P43351 1/20 0.37
PMP22 Q01453 1/20 0.37
NQO2 P16083 1/20 0.37
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
PDE4A P27815 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20170881 0.81 CYP1A2 (0.36) GAABCHEACHECYP3A4CYP1A2
SCHEMBL18473561 0.76 GAA (0.37) GAABCHEACHECYP3A4CYP1A2
SCHEMBL20170713 0.75 AGTR2 (0.41) PDE4APDE4BPDE4CPDE4D
SCHEMBL20170665 0.74 CYP3A4 (0.41) GAABCHEACHECYP3A4CYP1A2
SCHEMBL13301272 0.73 HTR1A (0.34) ACHE
SCHEMBL26205690 0.70 BCHE (0.39) BCHEACHECYP3A4CYP1A2CYP2D6
SCHEMBL6260285 0.67 SRD5A1 (0.55) CYP3A4HSD17B10ALDH1A1KDM4EMAPT
SCHEMBL6249634 0.67 SRD5A1 (0.55) CYP3A4HSD17B10ALDH1A1KDM4EMAPT
SCHEMBL29885479 0.65 MAOA (0.54) BCHEACHECYP2D6HSD17B10HIF1A
SCHEMBL21081223 0.64 ACHE (0.34) GAABCHEACHECYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed