SCHEMBL20170731

SCHEMBL20170731

C=CCNC1Cc2ccc(OC)c3c2C2C1CCC(NCCC)C2O3

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 3/20 0.43
HTR1A P08908 14/20 0.41
DRD2 P14416 2/20 0.32
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20170880 0.92 HCRTR1 (0.45) HCRTR1HTR1A
SCHEMBL20170799 0.81 HCRTR1 (0.47) HCRTR1HTR1A
SCHEMBL20170650 0.81 HCRTR1 (0.44) HCRTR1HTR1A
SCHEMBL20852459 0.79 HTR1A (0.41) HCRTR1HTR1A
SCHEMBL10223933 0.75 HCRTR1 (0.45) HCRTR1HTR1A
SCHEMBL20852445 0.72 HTR1A (0.35) HTR1A
SCHEMBL20170738 0.68 HTR1A (0.40) HCRTR1HTR1ADRD2DRD4DRD3
SCHEMBL18473435 0.67 HCRTR1 (0.42) HCRTR1HTR1A
SCHEMBL13972295 0.66 HCRTR1 (0.41) HCRTR1HTR1ADRD2DRD4DRD3
SCHEMBL18473438 0.66 HCRTR1 (0.41) HCRTR1HTR1ADRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed