SCHEMBL20170650

SCHEMBL20170650

CN[C@H]1Cc2ccc(OC)c3c2C2[C@H](O3)C(NCCO)CC[C@@H]21

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 5/20 0.44
HTR1A P08908 1/20 0.32
ADRA2A P08913 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30
ADRA1D P25100 1/20 0.30
ADRA1A P35348 1/20 0.30
ADRA1B P35368 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20170880 0.89 HCRTR1 (0.45) HCRTR1HTR1A
SCHEMBL10223933 0.82 HCRTR1 (0.45) HCRTR1HTR1A
SCHEMBL20170738 0.81 HTR1A (0.40) HCRTR1HTR1AADRA1B
SCHEMBL20170731 0.81 HCRTR1 (0.43) HCRTR1HTR1A
SCHEMBL20170692 0.73 HCRTR1 (0.36) HCRTR1HTR1AADRA1A
SCHEMBL20170822 0.71 OPRM1 (0.51)
SCHEMBL20170799 0.71 HCRTR1 (0.47) HCRTR1HTR1A
SCHEMBL13072367 0.70 OPRM1 (0.34) HCRTR1
SCHEMBL20170820 0.68 HCRTR1 (0.46) HCRTR1
SCHEMBL20170646 0.66 OPRM1 (0.42) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed