SCHEMBL20170799

SCHEMBL20170799

C=CCNC1Cc2ccc(OC)c3c2C2C1CCC(OC(C)=O)C2O3

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 5/20 0.47
HTR1A P08908 8/20 0.42
GABRA1 P14867 2/20 0.34
GABRB2 P47870 2/20 0.34
NQO2 P16083 1/20 0.31
MTNR1A P48039 1/20 0.31
MTNR1B P49286 1/20 0.31
OPRK1 P41145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20170880 0.82 HCRTR1 (0.45) HCRTR1HTR1A
SCHEMBL20170731 0.81 HCRTR1 (0.43) HCRTR1HTR1A
SCHEMBL20170753 0.74 GABRA1 (0.39) HCRTR1GABRA1GABRB2NQO2MTNR1A
SCHEMBL20170650 0.71 HCRTR1 (0.44) HCRTR1HTR1A
SCHEMBL18473438 0.64 HCRTR1 (0.41) HCRTR1HTR1AOPRK1
SCHEMBL13972295 0.64 HCRTR1 (0.41) HCRTR1HTR1AOPRK1
SCHEMBL13972294 0.64 HCRTR1 (0.41) HCRTR1HTR1AOPRK1
SCHEMBL20170820 0.64 HCRTR1 (0.46) HCRTR1OPRK1
SCHEMBL20170592 0.63 MTNR1A (0.40) HCRTR1NQO2MTNR1AMTNR1B
SCHEMBL20170750 0.63 OPRM1 (0.51) GABRA1GABRB2OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed