SCHEMBL20170784

SCHEMBL20170784

COc1ccc2c(c1O)[C@]13CC(=O)CCC1C1NCC21C3

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.51
KDM4E B2RXH2 1/20 0.35
CYP3A4 P08684 1/20 0.35
MAPT P10636 1/20 0.35
CYP2D6 P10635 1/20 0.35
MRGPRX2 Q96LB1 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
OPRD1 P41143 5/20 0.33
OPRM1 P35372 3/20 0.33
OPRK1 P41145 2/20 0.33
PDE4A P27815 2/20 0.33
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20170840 0.81 GAA (0.41) GAAKDM4EMAPT
SCHEMBL20170807 0.76 GAA (0.48) GAACYP3A4CYP2D6OPRD1OPRM1
SCHEMBL10222582 0.72 GAA (0.66) GAAKDM4ECYP3A4MAPTCYP2D6
SCHEMBL14768978 0.72 GAA (0.66) GAAKDM4ECYP3A4MAPTCYP2D6
SCHEMBL21091196 0.70 GAA (0.61) GAAKDM4ECYP3A4MAPTCYP2D6
SCHEMBL18878794 0.69 GAA (0.68) GAAKDM4ECYP3A4MAPTCYP2D6
SCHEMBL18994724 0.68 GAA (0.67) GAAKDM4ECYP3A4MAPTCYP2D6
SCHEMBL12717590 0.67 GAA (1.00) GAAKDM4ECYP3A4MAPTCYP2D6
SCHEMBL12960964 0.67 GAA (1.00) GAAKDM4ECYP3A4MAPTCYP2D6
SCHEMBL21148321 0.67 GAA (1.00) GAAKDM4ECYP3A4MAPTCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed